Fa'amatalaga o oloa
Artesunate e faia mai le artemisinin vaega aoga na maua mai Artemisia annua, lea e tulaga ese i Saina, e ala i le faʻaogaina o vailaʻau.E masani lava ona galue i luga ole vaega mumu clones o malaria parasites.E na'o le pau lea o le mea e maua mai ai le artemisinin e mafai ona faia i ni sauniuniga solu vai i le taimi nei.E mafai ona fasiotia le Plasmodium i le vaega erythrocytic ma ausia ai le aafiaga antimalarial.O loʻo i ai uiga o le maualuga o le antimalarial, vave antipyretic, taimi puʻupuʻu mo le suiga le lelei o Plasmodium, ma aʻafiaga laiti oona ma itu.O le filifiliga muamua lea mo togafitiga o le malaria ogaoga.
1. La'au tupuaga
O le Artesunate o se mea e maua mai i le artesunate semi synthetic.
2. Mechanism of action
Le faiga ole gaioiga ole artemisinin artesunate.E muamua galue i luga o le meaʻai vesicle membrane, surface membrane ma mitochondria o Plasmodium.O le lona lua o le membrane faaniukilia ma le endoplasmic reticulum.E le gata i lea, e iai foi se aafiaga patino i le chromatin i totonu o le nucleus.A o galue muamua lenei oloa i luga o le paʻu o meaʻai, ma taofia ai le faʻaogaina o meaʻai, o le malaria parasite e vave matelaina i amino acids, faʻavavevave ona fausia vesicles autophagic, ma faʻaauau ona alu ese mai le tino, ma le tele o le cytoplasm ma mate.
3. Matafaioi
1. Vailaau fa'ama'i
O le Artesunate ose vaila'au fa'atosina e masani ona fa'aaogaina.O se mea e maua mai i le artesunate ma sesquiterpene lactone structure, o se faʻaititia o le artesunate.
2. O a'afiaga fa'ama'i fa'ama'i
O le Artesunate e iai sona aafiaga taua i luga o sela tumo ma e le faigofie ona maua ai le tetee atu i fualaau.I tausaga talu ai nei, ua iloa ai e le au sikola i le fale ma fafo atu e mafai e le artesunate ona faia se matafaioi anti-tumour e ala i le taofiofia o le tuputupu aʻe o le tumo, faʻaosofia le eseesega o le tumo ma le apoptosis, faʻatonutonuina le faʻaliliuina o faailoilo o le cell, faʻafefe angiogenesis tumo, faʻalavelave osofaʻiga ma metastasis, sensitizing anti. -tumor chemotherapy vailaʻau ma faʻafoʻisia teteʻe fualaau.
4, fanua talosaga
1. Alamanuia tau vailaau
Fua Fa'atatau
FA'ATA'IGA O KAMUMU | |
Igoa Oloa | Artesunate |
CAS | 88495-63-0 |
Fuainumera Fa'ainumera | C19H28O8 |
Brand | Hande |
Mtagata gaosi oloa | Yunnan Hande Bio-Tech Co., Ltd. |
Catunuu | Kunming,China |
Fa'atuina | 1993 |
BASIC FAAMATALAGA | |
Synonyms | ARTENSUNATE;Butanedioicacid,1-[(3R,5aS,6R,8aS,9R,10S,12R,12aR)-decahydro-3,6,9-trimethyl-3,12-epoxy-12H-pyrano[4,3-j ]-1,2-benzodioxepin-10-yl]ester;Artesunate(3R,5aS,6R,8aS,9R,10S,12R,12aR)-Decahydro-3,6,9-trimethyl-3,12-epoxy-12H -pyrano(4,3-j)-Chemicalbook1,2-benzodioxepin-10-olhydrogensuccinate;ARTESUNATE;ArtesunateC19H28O8;Artemisininmonosuccinate;ArtesunicAcid;ButanedioicAcidMono(3R,5aS,6R,8aS,9R,10R2aS,12,10R2aS,12,10R2aS,12R,10R2aS,12R,10R2aS ,6,9-trimethyl-3,12-epoxy-12H-pyrano[4,3-j]-1,2-benzodioxepin-10-yl]Ester |
Fauga | |
mamafa | 384.42 |
HS Code | N/A |
Tulaga leleiSfa'amatalaga | Kamupani Fa'amatalaga |
Ctusi faamaonia | N/A |
Su'ega | Fa'apitoa e tusa ai ma mana'oga o tagata fa'atau |
Fa'aaliga | tioata paepae |
Auala o le Aveina | Artemisia annua Linn. |
Mafai Faaletausaga | Fa'apitoa e tusa ai ma mana'oga o tagata fa'atau |
afifi | Fa'apitoa e tusa ai ma mana'oga o tagata fa'atau |
Metotia Su'ega | HPLC |
Logistics | Fa'atelefelauaigas |
PmanuiaTerms | T/T, D/P, D/A |
Oisi | Talia su'etusi a tagata faatau i taimi uma;Fesoasoani i tagata fa'atau ile resitalaina o tulafono faatonutonu. |
Fa'amatalaga o oloa a Hande
1. O oloa uma na fa'atauina e le kamupani o mea fa'amea fa'ato'a mae'a.O oloa o lo'o fa'atatau tonu lava i tagata gaosi oloa o lo'o i ai agava'a fa'apitoa, ma o mea mata'ina e le o ni oloa fa'ai'uga.
2. Ole aoga fa'apitoa ma fa'aoga o lo'o a'afia i le fa'atomuaga e maua uma mai tusitusiga fa'asalalau.E le fautuaina e tagata taʻitoʻatasi le faʻaogaina saʻo, ma e teena faʻatauga a le tagata lava ia.
3. O ata ma faʻamatalaga o oloa i luga o lenei upega tafaʻilagi e mo naʻo faʻamatalaga, ma o le oloa moni e tatau ona manumalo.
Hande falegaosimea:
Yunnan hande Biotechnology Co., Ltd., na faavaeina ia Aokuso 1993, o se atinaʻe faʻatekonolosi maualuga faʻapitoa i suʻesuʻega ma atinaʻe biotechnology.A maeʻa tausaga o atinaʻe, ua faʻavaeina e le hande se faiga lelei atoatoa, pulea le lelei o oloa e tusa ai ma tulaga maualuga, ma faʻateleina le tau o le gaosiga o gafatia.O ana oloa ua pasia le faʻamaonia o tulafono ma tulafono faʻavaomalo, ma avea ma se gaosiga o mea faʻapitoa e faʻamalieina ai tagata uma.
Avea ma tagata sili ona lelei e tuʻuina atu mea mataʻutia ma atinaʻe ma le faʻamaoni!
Faʻafeiloaʻi e faʻafesoʻotaʻi aʻu e ala i le lafoina o imeli imarketing@handebio.com